5-amino-1MQ

Also: 5-amino-1-methylquinolinium, 5A1MQ

Summary

5-amino-1MQ is not a peptide. It is a small molecule that inhibits nicotinamide N-methyltransferase, an enzyme that sits between cellular metabolism and the regulation of gene activity. It is a research compound with no published human data at all, and it is on this site because listed suppliers sell it alongside peptides.

What it targets

The enzyme this compound blocks methylates nicotinamide using the body's universal methyl donor, which links one-carbon metabolism to NAD+ levels; a 2024 review describes how differently it behaves across tissues and surveys its reported roles in cancer, liver, brain, lung, cardiovascular and kidney disease, which is a reason to expect effects beyond fat tissue. The most direct evidence for the compound itself is a 2024 study in which mice made obese on a high-fat diet received it daily for 28 days: the authors report dose-dependent limits on body weight and fat gain, better glucose tolerance and insulin sensitivity, lower insulin levels and reduced fatty-liver changes, alongside measurements of how the compound behaves after intravenous, oral and subcutaneous administration. Earlier work validated the enzyme as a target, including a related inhibitor whose effects disappeared in mice lacking the enzyme. Every result above is in mice or cells.

body weight and fat mass in diet-induced obese miceglucose tolerance and insulin sensitivity in micefatty-liver changes in micethe enzyme as a metabolic drug target (review and cell work)

Clinical Research

Nicotinamide N-methyltransferase inhibition mitigates obesity-related metabolic dysfunction
Babula JJ, Bui D, Stevenson HL, et al. (2024). Diabetes, Obesity and Metabolism. animal diet-induced obese mice given the compound daily for 28 days, plus pharmacokinetic work after intravenous, oral and subcutaneous administration
Selective and membrane-permeable small molecule inhibitors of nicotinamide N-methyltransferase reverse high fat diet-induced obesity in mice
Neelakantan H, Vance V, Wetzel MD, et al. (2018). Biochemical Pharmacology. animal cultured adipocytes and permeability assays, then mice made obese on a high-fat diet
A small molecule inhibitor of Nicotinamide N-methyltransferase for the treatment of metabolic disorders
Kannt A, Rajagopal S, Kadnur SV, et al. (2018). Scientific Reports. animal diet-induced obese mice, ob/ob and db/db mice, and NNMT knockout mice as a specificity control
Exploring NNMT: from metabolic pathways to therapeutic targets
Park J, Shin EJ, Kim TH, et al. (2024). Archives of Pharmacal Research. review n/a (review)

All research on 5-amino-1MQ →

Suppliers stocking 5-amino-1MQ

11 of the 30 listed suppliers. Each row opens its full listing.

Aussie Peptides Australia Research use only. Statements have not been evaluated by the TGA. We do not ship internationally at this time. Australian Peptide Site Australia Intended for laboratory and scientific research use only. BioLongevity Labs United States All products are manufactured for research use only. Research Use Only products sold here are intended solely for laboratory research. HEEZ Research United States All products are for laboratory developmental research use only. Products are not for human consumption. HEEZ Research is a chemical supplier. Midshire Labs United Kingdom All Midshire Labs products are sold strictly for research purposes only. They are not intended for human consumption, medical, veterinary, or diagnostic use. Nationwide Peptides United States For Research Use Only. Products are not intended for human or animal consumption, ingestion, injection, or any form of administration. Peak Lab Peptides United States All products on this site are for research and development use only. Products are not for human consumption of any kind. Protide Health United States All products are supplied for laboratory research only and are not for human or animal consumption, medical use, veterinary use, or any therapeutic, diagnostic, or clinical purpose. Pure Peptides UK United Kingdom All products are for research use only. Synapse Peptides Australia Australia All products are supplied strictly for research purposes only and are not intended for human or veterinary use. XL Peptides United Kingdom All products are exclusively sold for research purposes. They are not intended for human use, therapeutic, diagnostic, or clinical application.