Epitalon

Also: epithalon, epithalone, AEDG peptide, Ala-Glu-Asp-Gly

Summary

Epitalon is a synthetic four-amino-acid peptide (Ala-Glu-Asp-Gly) designed from the amino acid composition of epithalamin, an extract of the bovine pineal gland. It comes from the same Russian bioregulator programme as several other peptides on this site. Twenty-five years of published work is in cells, animals and computer models; there is no human trial among the papers linked here.

What it targets

The claim most often attached to epitalon comes from a short 2003 report in which adding the peptide to cultured human fetal fibroblasts, cells that do not normally make telomerase, was said to switch the enzyme on and lengthen telomeres. That is a cell-culture finding; the paper's suggestion that it could extend the lifespan of an organism is not demonstrated in it. In mice bred to develop mammary tumours, monthly courses of epitalon were associated with fewer and smaller tumours and lower HER-2/neu gene expression, while a similar short peptide tested alongside it had the opposite effect. In mouse egg cells aged in culture, epitalon reduced reactive oxygen species and markers of deterioration. A 2025 independent review collects this work, notes reported effects on melatonin synthesis and several enzymes, and says it remains uncertain whether these are the only mechanisms involved.

telomerase activity in cultured human cellsspontaneous mammary tumours in transgenic miceegg cell deterioration in culturemelatonin and enzyme activity (reviewed)

Clinical Research

Overview of Epitalon - Highly Bioactive Pineal Tetrapeptide with Promising Properties
Araj SK, Brzezik J, Madra-Gackowska K, Szeleszczuk L (2025). International Journal of Molecular Sciences. review n/a (review of 25 years of in vitro, animal and computational work)
Epithalon Peptide Induces Telomerase Activity and Telomere Elongation in Human Somatic Cells
Khavinson VK, Bondarev IE, Butyugov AA (2003). Bulletin of Experimental Biology and Medicine. in-vitro cultured human fetal fibroblasts, a cell type that does not normally express telomerase
Inhibitory effect of the peptide epitalon on the development of spontaneous mammary tumors in HER-2/neu transgenic mice
Anisimov VN, Khavinson VK, Provinciali M, et al. (2002). International Journal of Cancer. animal female HER-2/neu transgenic mice, treated monthly from 2 months of age, against saline and a comparison peptide
Epitalon protects against post-ovulatory aging-related damage of mouse oocytes in vitro
Yue X, Liu SL, Guo JN, et al. (2022). Aging. in-vitro mouse oocytes aged in culture for 6, 12 and 24 hours after ovulation

All research on Epitalon →

Suppliers stocking Epitalon

12 of the 30 listed suppliers. Each row opens its full listing.

Au Peptide Labs Australia For laboratory research use only. Not for human consumption. Aussie Peptides Australia Research use only. Statements have not been evaluated by the TGA. We do not ship internationally at this time. Australian Peptide Site Australia Intended for laboratory and scientific research use only. Imperial Peptides UK United Kingdom In Vitro Research Use Only. Not for human or veterinary consumption. Licensed Peptides United States Supplied strictly for laboratory research use only. Not intended for human consumption, veterinary use, therapeutic applications, or diagnostic use. No dosing instructions are provided. Nationwide Peptides United States For Research Use Only. Products are not intended for human or animal consumption, ingestion, injection, or any form of administration. Pept Australia Products sold by Pept are intended for laboratory research purposes only and are not approved for human consumption. Protide Health United States All products are supplied for laboratory research only and are not for human or animal consumption, medical use, veterinary use, or any therapeutic, diagnostic, or clinical purpose. Pure Peptides UK United Kingdom All products are for research use only. Synapse Peptides Australia Australia All products are supplied strictly for research purposes only and are not intended for human or veterinary use. UK Peptides United Kingdom All products are sold exclusively for in-vitro research. They are not for human or veterinary use. XL Peptides United Kingdom All products are exclusively sold for research purposes. They are not intended for human use, therapeutic, diagnostic, or clinical application.